Foundations · Section 10 of 117

Functional groups

Practice this — interactive lesson

A functional group is a small, specific arrangement of atoms that behaves the same way whichever molecule it is bolted onto. An O–H on a two-carbon chain and an O–H on a thirty-carbon steroid do the same chemistry, at roughly the same rate, with the same reagents. That is why organic chemistry is organized around groups rather than around molecules: there are tens of millions of known compounds and only a few dozen groups, and the group is what a molecule does.

The rest of the molecule — the carbon chain or ring the group sits on — is a spectator. The previous section explains why. A C–C bond joins two atoms of identical electronegativity (2.55 against 2.55), and a C–H bond is close enough (2.55 against 2.20) that the difference does not matter. Neither has a δ+ end worth attacking, and neither carries a lone pair to attack with. Every bond in a functional group, by contrast, is either polar, or a lone pair, or a π bond sitting exposed above and below the plane of the atoms. The group is where the electrons are uneven or accessible; the skeleton is where they are not.

Read a structure by looking for anything that is not C–C or C–H: an oxygen, a nitrogen, a halogen, a sulfur, or a double or triple bond. Circle each one. Those circles are the functional groups, and for the rest of the course they are the only parts of the molecule you will be asked about.

The groups this course uses

Nineteen groups cover essentially everything in a first-year course. The structures below are drawn in condensed and Lewis form — R stands for any carbon chain, and R′ for a second one that need not match. The naming column is a preview: how a group shows up in a compound's name is the business of IUPAC Nomenclature, and you do not need it yet. It is here because the suffix is often the fastest way to recognize the group in a name you meet on a label.

GroupStructureName previewAn example you have met
AlkaneC–C and C–H bonds only, CH3CH2CH3suffix -anePropane, the gas in a camping stove
AlkeneC=C, CH2=CH2suffix -eneEthylene, the hormone that ripens fruit
AlkyneC≡C, HC≡CHsuffix -yneAcetylene, the fuel in a welding torch
Alkyl halideR–X (X = F, Cl, Br, I), CH2Cl2prefix fluoro-, chloro-, bromo-, iodo-Dichloromethane, the solvent in paint stripper
AlcoholR–OH, CH3CH2OHsuffix -olEthanol
EtherR–O–R′, CH3CH2OCH2CH3prefix alkoxy- (methoxy-, ethoxy-)Diethyl ether, the first surgical anesthetic
AmineR–NH2, R2NH or R3N; (CH3)3Nsuffix -amine, prefix amino-Trimethylamine, the smell of fish
ThiolR–SH, CH3CH2SHsuffix -thiolEthanethiol, added to natural gas so a leak can be smelled
AldehydeR–CH=O, written RCHO; CH3CHOsuffix -alAcetaldehyde, what ethanol becomes in the liver
KetoneR–C(=O)–R′, written RCOR′; CH3COCH3suffix -oneAcetone, nail-polish remover
Carboxylic acidR–C(=O)–OH, written RCOOH; CH3COOHsuffix -oic acidAcetic acid, vinegar
EsterR–C(=O)–OR′, written RCOOR′; CH3COOCH2CH3suffix -oate, two words: ethyl acetateEthyl acetate, the pear-drop smell of nail polish
AmideR–C(=O)–NH2, NHR′ or NR′2; CH3CONH2suffix -amideAcetaminophen; the peptide bond in every protein
Acid chlorideR–C(=O)–Cl, written RCOCl; CH3COClsuffix -oyl chlorideAcetyl chloride — a lab reagent, too reactive toward water to be sold in a shop
AnhydrideR–C(=O)–O–C(=O)–R, (CH3CO)2Osuffix -oic anhydrideAcetic anhydride, the reagent that turns salicylic acid into aspirin
NitrileR–C≡N, CH2=CHCNsuffix -nitrile, prefix cyano-Acrylonitrile, spun into acrylic sweaters
Aromatic ringC6H6 benzene, or C6H5– as a substituentparent benzene, prefix phenyl-Toluene, C6H5CH3, in paint thinner
Phenolan OH directly on an aromatic ring, C6H5OHparent phenolThe active part of many antiseptics
Nitro groupR–NO2, drawn R–N+(=O)–Oprefix nitro- (it is never the suffix)TNT, trinitrotoluene, CH3C6H2(NO2)3

Two rows deserve a second look with the previous sections in hand. The nitro group's nitrogen has four bonds, so it carries a formal charge of +1, and the singly bonded oxygen carries −1: that is the formal-charge arithmetic from earlier in this chapter, and a nitro group drawn with a neutral four-bonded nitrogen is the five-bonded-carbon error in disguise. And the amine row lists three structures rather than one, because the nitrogen can carry one, two or three carbons and still be an amine — which matters below.

The carbonyl family: what is attached to the C=O

AldehydeORHCδ+δ−attached: HKetoneORR′Cδ+δ−attached: a second carbonCarboxylic acidOROHCδ+δ−attached: OHEsterOROR′Cδ+δ−attached: O–carbonAmideORNH₂Cδ+δ−attached: N (NH₂, NHR′ or NR′₂)Acid chlorideORClCδ+δ−attached: ClAnhydrideOORROCCδ+δ−attached: O that leads to a second C=OThe C=O is the same in all seven: carbon δ+, oxygen δ− with two lone pairs.Only the atom on the right changes, and it is the whole name.
Seven groups, one carbonyl. Find the C=O, then read the atom on its right: H, a carbon, OH, OR′, N, Cl, or an oxygen that continues to another C=O. That one atom is the entire difference between an aldehyde and an ester, and it is what every "identify the functional group" question is really asking.The polar bond is marked identically in every panel because it is identical in every one: the carbonyl carbon is the most electron-poor carbon in the whole table, for the electronegativity reason of the previous section, doubled by the second bond to oxygen. What the right-hand atom changes is not whether that carbon is attacked but what happens afterward, which is the story of three later chapters.

Seven of the groups in the table contain a carbonyl, a carbon double-bonded to oxygen, and they are the seven most confused. The distinction is mechanical once you know where to look: find the C=O, then read the other two things attached to its carbon. One of them is usually carbon or hydrogen; the other one names the group.

Attached to the C=O carbonGroupCondensed
H (and a carbon, or a second H)AldehydeRCHO
Carbon on both sidesKetoneRCOR′
OHCarboxylic acidRCOOH
O–carbon (OR′)EsterRCOOR′
NAmideRCONH2, RCONHR′, RCONR′2
ClAcid chlorideRCOCl
O attached to a second C=OAnhydrideRCO–O–COR

The single most tested recognition skill in the course is that table, read in reverse: given a structure, say which row it is. Practice it on the condensed formulas until RCOOR′ and RCOR′ look as different to you as they do to a chemist.

Worked example — three formulas that differ by one atom

CH3COCH3. The C=O carbon is bonded to CH3 and CH3: carbon on both sides, so a ketone (acetone).

CH3COOCH3. Same start, but now there is an oxygen between the carbonyl and the second methyl. One side carbon, the other side O–C, so an ester (methyl acetate). The extra O is the whole difference, and it is the atom people skip when reading quickly.

CH3OCH3. No C=O at all: an oxygen with a carbon on each side is an ether. An ester is an ether-like O plus a carbonyl on one side; an ether has the O alone.

Primary, secondary, tertiary

Several groups are further classified by degree of substitution, and the rule has two versions.

For a carbon, count the other carbons bonded to it: one is primary (1°), two is secondary (2°), three is tertiary (3°), four is quaternary (4°). Alcohols and alkyl halides take the degree of the carbon that carries the OH or the halogen. CH3CH2OH is a primary alcohol; (CH3)2CHOH is secondary; (CH3)3COH is tertiary. Same for CH3CH2Br, (CH3)2CHBr and (CH3)3CBr.

For an amine, count the carbons bonded to the nitrogen, not to any carbon. CH3NH2 is primary, (CH3)2NH is secondary, (CH3)3N is tertiary. The reason for the different rule is that the nitrogen is the reactive atom, and what matters about it is how crowded it is.

The exam trap. (CH3)3C–OH is a tertiary alcohol; (CH3)3C–NH2 is a primary amine. Same tert-butyl carbon in both. The alcohol is classified by that carbon, which has three carbon neighbors; the amine is classified by its nitrogen, which has one. If a question puts a bulky carbon next to an NH2, it is asking exactly this.

Why polarity tells you where a group will react

The previous section said a polar bond has a δ+ end and a δ− end, and the section before it gave the numbers. Put them against the table above and a pattern falls out.

Here is the preview, and it is the one to hang everything on. Every group has either an electron-rich site — a lone pair, a π bond, a δ− atom — or an electron-poor one, a δ+ carbon, and most have both. Organic Structure & Electron Movement will name those sites nucleophiles and electrophiles, and every reaction after that is an electron-rich site finding an electron-poor one. Nothing about the reactions is being taught here. What is being taught is that you can already see, from electronegativity alone, where on each group they will happen.

Common mistakes

Worked examples: real molecules, every group named

Worked example — aspirin, HOOC–C6H4–O–CO–CH3

Find the non-alkane pieces. A C6H4 unit, a COOH, and an O–CO–CH3.

C6H4 with two things attached is a benzene ring carrying two substituents: an aromatic ring.

HOOC– is a C=O with an OH on it: a carboxylic acid. Its other neighbor is a ring carbon.

–O–CO–CH3 is the one to read slowly. There is a C=O; one side of it is CH3, the other side is an oxygen that continues to a carbon (the ring). Carbon on one side, O–C on the other: an ester. It is not an ether, because the O sits next to a carbonyl, and the C=O is not a ketone, because one of its neighbors is oxygen.

Three groups: aromatic ring, carboxylic acid, ester. The two-carbon CH3CO fragment is the acetyl group, which is what the "a" in aspirin and the "acet" in acetylsalicylic acid refer to.

Worked example — acetaminophen, HO–C6H4–NH–CO–CH3

The ring is again an aromatic ring with two substituents.

HO– on the ring. The OH is directly on an aromatic carbon, so this is a phenol, not an alcohol. (Same atoms as an alcohol, different group, and a different chemistry.)

–NH–CO–CH3. The nitrogen is bonded to a C=O. That makes it an amide, not an amine. Read the carbonyl too: its neighbors are N and CH3, and the N is the one that names it. It is not a ketone, and there is no amine anywhere in the molecule.

Two groups plus a ring: phenol and amide. A student who writes "alcohol, amine, ketone" has found all the right atoms and named all three groups wrongly, which is why this molecule is a favorite on exams.

Worked example — ibuprofen, (CH3)2CHCH2–C6H4–CH(CH3)–COOH

Left of the ring: (CH3)2CHCH2– is carbon and hydrogen only, an isobutyl chain. Alkane, spectator. Notice how much of the molecule that is.

The ring: aromatic, two substituents.

Right of the ring: –CH(CH3)–COOH. The COOH is a carboxylic acid. The CH that carries it is bonded to three carbons (the methyl, the ring, and the carboxyl carbon), so that carbon is tertiary, a detail that matters later for its stereochemistry.

One aromatic ring, one carboxylic acid, and a lot of spectator. Ibuprofen, aspirin and acetaminophen are all painkillers, and the only group the three share is the aromatic ring. What they do in the body has more to do with the acid, the ester and the amide respectively than with the ring, which is the point of the section.

What carries forward

All of it, in three directions. Organic Structure & Electron Movement redraws these groups in skeletal notation, which hides the spectator carbons so that the groups stand out even more, and then names the electron-rich and electron-poor sites you have just located. IUPAC Nomenclature turns the preview column of the table into a system, including what to do when one molecule has several groups. And from Acids & Bases onward, every chapter is titled after one of these rows.