Oxidation & Reduction · Section 62 of 116

Oxidizing alcohols

Practice this — interactive lesson

A primary alcohol can be oxidized to an aldehyde or straight past it to a carboxylic acid, and the aldehyde is very often the thing you actually want. Learning this section is learning which reagent stops where, and the reason turns out to be a single mechanistic detail: whether there is water in the flask.

What each class of alcohol can become

SubstrateMild oxidantStrong / aqueous oxidant
Primary alcoholAldehydeCarboxylic acid
Secondary alcoholKetoneKetone
Tertiary alcoholNo reactionNo reaction

The secondary column is the reassuring one: a ketone has no hydrogen left on the carbonyl carbon, so it cannot be oxidized further under these conditions and both reagents give the same thing. The choice of reagent only matters for primary alcohols.

Why water decides where a chromium oxidation stops

Chromium(VI) reagents oxidize an alcohol by way of a chromate ester, which then loses the carbinol C–H to give the carbonyl. For a primary alcohol that gives an aldehyde — and an aldehyde in water is in equilibrium with its hydrate, the gem-diol formed by water adding across the C=O.

That hydrate is, structurally, an alcohol again: it has an OH and a hydrogen on the same carbon. So the chromium reagent oxidizes it a second time, and the product is the carboxylic acid. Take the water away and the hydrate never forms, so the oxidation has nothing left to grip and stops at the aldehyde.

This is the whole explanation for the reagent list below. Anhydrous chromium reagent → aldehyde. Aqueous chromium reagent → carboxylic acid. It is not about strength, and adding less oxidant or shortening the reaction time does not reliably stop an aqueous oxidation at the aldehyde.

The reagents worth knowing

ANHYDROUS — PCC, Swern, DMPR–CH₂OH[O]no waterR–CHOno water, so no hydrate — nothing left to gripstops at the aldehydeAQUEOUS — Jones, CrO₃/H₂SO₄R–CH₂OH[O]R–CHO+ H₂OOHOHRHCthe hydrate: an OH and an H on one carbon — an alcohol again[O] againR–CO₂Hcarboxylic acidSame oxidant, same substrate, same carbinol C–H.The water is the entire difference.
Why a chromium oxidation stops in one flask and not in the other. Both runs make the aldehyde first; only in water does that aldehyde turn back into something carrying an OH and a hydrogen on the same carbon — which is exactly what the oxidant attacked the first time.The hydrate is never isolated and never appears in the answer, which is why this step is so easy to miss, and it is the reason the rule is about water rather than about strength. Using less Jones reagent or a shorter reaction time does not reliably stop the oxidation at the aldehyde, because the hydrate forms as fast as the aldehyde does. The Swern and DMP reach the same aldehyde by a route with no water anywhere in it.

Group them by outcome rather than by chemistry and the list is short: PCC, Swern and DMP give aldehydes; Jones and other aqueous Cr(VI) give carboxylic acids; all of them give ketones from secondary alcohols and nothing from tertiary ones.

Chromium reagents are toxic and environmentally nasty, which is why the Swern and DMP exist and why modern papers usually avoid chromium. Exams still ask about PCC and Jones constantly, so you need both — but it is worth knowing the metal-free options are not merely alternatives, they are the ones a working lab reaches for first.
Worked example — choosing by what must survive

You need to convert the primary alcohol of a molecule that also contains a secondary alcohol elsewhere, and you want the aldehyde.

Reagent choice. PCC, Swern or DMP will all stop at the aldehyde. None of them distinguishes a primary alcohol from a secondary one, though, so the secondary alcohol will be oxidized to a ketone at the same time.

The real answer is that you cannot solve this by reagent choice alone. You protect the secondary alcohol first, oxidize, then deprotect. Recognizing that a selectivity problem needs a protecting group rather than a cleverer oxidant is the actual skill being tested.

Oxidation levels, again

Read the whole section against the ladder from the last one and it compresses. An alcohol sits at one rung, an aldehyde or ketone one rung up, a carboxylic acid one rung above that. A primary alcohol has two rungs available because it has two hydrogens on the carbinol carbon; a secondary alcohol has one; a tertiary alcohol has none and therefore cannot climb at all.

What carries forward

Every one of these reactions runs backwards in the next section, where hydride reagents take carbonyls back down to alcohols. Holding both directions at once is what makes synthesis planning possible — a primary alcohol and an aldehyde are one oxidation apart in either direction, so a route that needs one from the other is a single step, and knowing which reagent gets you there without overshooting is the content.